what is the pharmacophore of the antiviral drug nevirapine ?
Homework Answers
Pharmacophore of any drug is the active part of the molecular that is responsible for its biological or pharmacological effects. Nevirapine structure has a hydrogen bond acceptor, hydrogen bond donor, hydrophobic atom/group, aromatic ring center and direction, nonaromatic ring center and direction, negatively charged group center, and positively charged group center. Each of these have different effects and can be easily identified on the structure of molecule. Other drugs with similar pharmacophore include erlotinib and zanamivir among many others.
D. Antiviral E. Antifungal 14. What type of drug is Metronidazole? A. Antibacterial, targets cell wall...
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1. Remdesivir is an antiviral drug that was developed as a treatment for the Ebola virus...
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The patient being treated with the antiviral agent amantadine. While the patient is receiving the drug, the np should mo...
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Chapter 40 Acyclovir Valacyclovir Anti-herpetic antiviral (synthetic nucleoside analogue) Amantadine (not commonly used) Oseltamivir Anti-influenza antiviral...
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As group, construct a table listing common classes of antiviral drugs ( agents for influenza A...
As group, construct a table listing common classes of antiviral drugs ( agents for influenza A and respiratory viruses, agents for herpes and CMV, agents for HIV/AIDS, and topical agents). Label columns for therapeutic actions, pharmacokinetics, contraindications, common adverse reactions, and important drug-drug interactions. Complete the table for each antiviral group. Pharmacology
(26 points) Kineties of an Antiviral Drug. In 2016, Nature reported the discovery of a small...
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Summarize the mode of action of major groups of antimicrobial and antiviral drugs. Summarize practices that...
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The patient is a 22 year old female who is 16 weeks pregnant and is scheduled...
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D. Antiviral E. Antifungal 14. What type of drug is Metronidazole? A. Antibacterial, targets cell wall synthesis B. Antibacterial, targets ribosomes/protein synthesis C. Antibacterial, other D. Antiviral E. Antifungal 15. What type of drug is Daptomycin? A. Antibacterial, targets cell wall synthesis B. Antibacterial, targets ribosomes/protein synthesis C. Antibacterial, other D. Antiviral E. Antifungal 16. What type of drug is Amphotericin B? A. Antibacterial, targets cell wall synthesis B. Antibacterial, targets ribosomes/protein synthesis C. Antibacterial, other
1. Remdesivir is an antiviral drug that was developed as a treatment for the Ebola virus and the Marburg virus. It is currently in clinical trials as a treatment for COVID-19. NH2 LON HOOH remdesivir The following questions are about the boxed portion of remdesivir, drawn below as its own molecule. a) Fill in the boxes about the hybridization and orbitals of this heterocycle. What is the hybridization of this N? o What orbital does this lone pair occupy? What...
Chapter 40 Acyclovir Valacyclovir Anti-herpetic antiviral (synthetic nucleoside analogue) Amantadine (not commonly used) Oseltamivir Anti-influenza antiviral Drug Name Drug Class & Indication(s) Contraindications Common Adverse Effects Major Interactions Review instructions for applying topical How soon should anti-flu drugs be Nurse Considerations: (Examples: Age, renal/hepatic precautions, safety administration, lab monitoring, patient teaching)
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